Assay Detail
Binding
CHEMBL845440
Review assay metadata, readout intent, target linkage, and publication context from the same page.
The compound was evaluated for its inhibitory effect of dual specificity phosphatases of VHR
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and characterization of a potent and selective protein tyrosine phosphatase inhibitor, 2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.30 | 4.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL89067 | — | — | 1 | 4.30 |
| CHEMBL86473 | VANADATE | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL89067 | — | IC50 | = | 50200.0 | nM | 4.30 |
| CHEMBL86473 | VANADATE | IC50 | = | 105800.0 | nM | - |