Assay Detail
Binding
CHEMBL853710
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of TPA-induced NF-kappaB activity in HepG2 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HepG2 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and cancer chemopreventive activity of zapotin, a natural product from Casimiroa edulis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.12 | 5.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL375582 | ZAPOTIN | — | 1 | 5.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL375582 | ZAPOTIN | IC50 | = | 7600.0 | nM | 5.12 |