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Assay Detail

CHEMBL855657

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Superoxide anion radical scavenging activity by xanthine/xanthine oxidase method
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Free radical scavengers from the medicinal mushroom Inonotus xeranticus and their proposed biogenesis.
Lee IK, Jung JY, Seok SJ, Kim WG, Yun BS.
Bioorg Med Chem Lett (2006) 16 : 5621 -5624
PubMed 16908141 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.84 5.54

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL145 CAFFEIC ACID 3.0 1 5.54
CHEMBL222021 PROTOCATECHUALDEHYDE 1 4.60
CHEMBL448733 METHYLINOSCAVIN D 1 4.39
CHEMBL218276 INOSCAVIN D 1 -
CHEMBL3989727 VITAMIN E 4.0 1 -
CHEMBL37537 PROTOCATECHUIC ACID 1 -
CHEMBL218423 PHELLIGRIDIN D 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL145 CAFFEIC ACID IC50 = 2900.0 nM 5.54
CHEMBL222021 PROTOCATECHUALDEHYDE IC50 = 25300.0 nM 4.60
CHEMBL448733 METHYLINOSCAVIN D IC50 = 40700.0 nM 4.39
CHEMBL218276 INOSCAVIN D IC50 > 100000.0 nM -
CHEMBL3989727 VITAMIN E IC50 > 100000.0 nM -
CHEMBL37537 PROTOCATECHUIC ACID IC50 > 100000.0 nM -
CHEMBL218423 PHELLIGRIDIN D IC50 > 100000.0 nM -