Assay Detail
Functional
CHEMBL859007
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Antibacterial activity against Clavibacter michiganensis
8
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Clavibacter michiganensis |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
A minimalist design approach to antimicrobial agents based on a thionin template.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 8 | 6.29 | 7.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4299737 | — | — | 2 | 7.52 |
| CHEMBL269753 | — | — | 1 | 6.29 |
| CHEMBL412491 | — | — | 1 | 6.13 |
| CHEMBL372354 | — | — | 1 | 6.05 |
| CHEMBL219285 | — | — | 1 | 6.05 |
| CHEMBL373375 | — | — | 1 | 5.49 |
| CHEMBL219374 | — | — | 1 | 5.29 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4299737 | — | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL4299737 | — | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL269753 | — | EC50 | = | 510.0 | nM | 6.29 |
| CHEMBL412491 | — | EC50 | = | 740.0 | nM | 6.13 |
| CHEMBL372354 | — | EC50 | = | 900.0 | nM | 6.05 |
| CHEMBL219285 | — | EC50 | = | 900.0 | nM | 6.05 |
| CHEMBL373375 | — | EC50 | = | 3270.0 | nM | 5.49 |
| CHEMBL219374 | — | EC50 | = | 5130.0 | nM | 5.29 |