Assay Detail
Binding
CHEMBL860427
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [125I]LVA antagonist from human vasopressin 2 receptor expressed in HEK293-EBNA cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293-EBNA |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Discovery and development of a new class of potent, selective, orally active oxytocin receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.60 | 5.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1254117 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1254117 | — | Ki | = | 2500.0 | nM | 5.60 |