Assay Detail
Binding
CHEMBL861857
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Inhibition of LF
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bacillus anthracis |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
The discovery of a potent and selective lethal factor inhibitor for adjunct therapy of anthrax infection.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.27 | 7.27 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL204593 | — | — | 1 | 7.27 |
| CHEMBL514138 | CGS-27023A | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL204593 | — | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL514138 | CGS-27023A | IC50 | - | — | - |