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Assay Detail

CHEMBL863347

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [125I]-echistatin from alphavbeta3 integrin receptor
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 7 — Homologous single protein target
Curated By Autocuration

Target

Integrin alpha-V/beta-3 (CHEMBL1907598)
Type PROTEIN COMPLEX
Organism Homo sapiens

Publication

Grafting aminocyclopentane carboxylic acids onto the RGD tripeptide sequence generates low nanomolar alphaVbeta3/alphaVbeta5 integrin dual binders.
Casiraghi G, Rassu G, Auzzas L, Burreddu P, Gaetani E, Battistini L, Zanardi F, Curti C, Nicastro G, Belvisi L, Motto I, Castorina M, Giannini G, Pisano C.
J Med Chem (2005) 48 : 7675 -7687
PubMed 16302808 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 14 7.72 8.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL392303 1 8.85
CHEMBL556402 1 8.82
CHEMBL534934 1 8.34
CHEMBL557157 1 8.25
CHEMBL534713 1 8.14
CHEMBL540622 1 8.11
CHEMBL534712 1 8.00
CHEMBL429876 CILENGITIDE 3.0 1 7.72
CHEMBL534933 1 7.45
CHEMBL534711 1 7.35
CHEMBL539850 1 7.29
CHEMBL539338 1 6.88
CHEMBL411941 CYCLORGDFV 1 6.71
CHEMBL540618 1 6.15

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL392303 IC50 = 1.4 nM 8.85
CHEMBL556402 IC50 = 1.5 nM 8.82
CHEMBL534934 IC50 = 4.6 nM 8.34
CHEMBL557157 IC50 = 5.6 nM 8.25
CHEMBL534713 IC50 = 7.2 nM 8.14
CHEMBL540622 IC50 = 7.7 nM 8.11
CHEMBL534712 IC50 = 9.93 nM 8.00
CHEMBL429876 CILENGITIDE IC50 = 18.9 nM 7.72
CHEMBL534933 IC50 = 35.6 nM 7.45
CHEMBL534711 IC50 = 44.7 nM 7.35
CHEMBL539850 IC50 = 51.4 nM 7.29
CHEMBL539338 IC50 = 132.9 nM 6.88
CHEMBL411941 CYCLORGDFV IC50 = 195.9 nM 6.71
CHEMBL540618 IC50 = 712.7 nM 6.15