Assay Detail
Binding
CHEMBL867616
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Inhibition of PP2A
4
Total Activities
4
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of protein phosphatase 2C inhibitors by virtual screening.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Activity | 3 | - | - |
| IC50 | 1 | 4.30 | 4.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL99039 | — | — | 1 | 4.30 |
| CHEMBL206583 | — | — | 1 | - |
| CHEMBL162783 | — | — | 1 | - |
| CHEMBL87223 | AMINOQUINURIDE | 2.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL99039 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL206583 | — | Activity | - | — | - | |
| CHEMBL162783 | — | Activity | - | — | - | |
| CHEMBL87223 | AMINOQUINURIDE | Activity | - | — | - |