Assay Detail
Binding
CHEMBL867768
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Inhibition of Agrobacterium sp. beta-glucosidase
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Agrobacterium sp. |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Fluorescent glycosidase inhibiting 1,5-dideoxy-1,5-iminoalditols.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 6 | 6.25 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL206468 | AFEGOSTAT | 2.0 | 1 | 8.15 |
| CHEMBL208677 | — | — | 1 | 6.85 |
| CHEMBL205510 | — | — | 1 | 6.50 |
| CHEMBL207481 | — | — | 1 | 6.00 |
| CHEMBL205592 | — | — | 1 | 5.05 |
| CHEMBL307429 | DUVOGLUSTAT | 2.0 | 1 | 4.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL206468 | AFEGOSTAT | Ki | = | 7.0 | nM | 8.15 |
| CHEMBL208677 | — | Ki | = | 140.0 | nM | 6.85 |
| CHEMBL205510 | — | Ki | = | 320.0 | nM | 6.50 |
| CHEMBL207481 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL205592 | — | Ki | = | 9000.0 | nM | 5.05 |
| CHEMBL307429 | DUVOGLUSTAT | Ki | = | 12000.0 | nM | 4.92 |