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Assay Detail

CHEMBL867947

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against VeroE6 cells infected with SARS coronavirus
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Chlorocebus sabaeus
Cell Type Vero
Confidence 1 — Organism
Curated By Intermediate

Target

Vero (CHEMBL391)
Type CELL-LINE
Organism Chlorocebus sabaeus

Publication

Synthesis, crystal structure, structure-activity relationships, and antiviral activity of a potent SARS coronavirus 3CL protease inhibitor.
Yang S, Chen SJ, Hsu MF, Wu JD, Tseng CT, Liu YF, Chen HC, Kuo CW, Wu CS, Chang LW, Chen WC, Liao SY, Chang TY, Hung HH, Shr HL, Liu CY, Huang YA, Chang LY, Hsu JC, Peters CJ, Wang AH, Hsu MC.
J Med Chem (2006) 49 : 4971 -4980
PubMed 16884309 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.22 6.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL213054 1 6.22
CHEMBL20636 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL213054 IC50 = 600.0 nM 6.22
CHEMBL20636 IC50 - -