Assay Detail
Functional
CHEMBL868078
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against human CMV by luciferase reporter gene assay in HFF cells
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | HFF |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Discovery of a novel series of inhibitors of human cytomegalovirus primase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 6.14 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL385537 | — | — | 1 | 7.70 |
| CHEMBL385536 | — | — | 1 | 7.41 |
| CHEMBL438246 | — | — | 1 | 6.77 |
| CHEMBL214960 | — | — | 1 | 6.72 |
| CHEMBL385412 | — | — | 1 | 6.26 |
| CHEMBL385156 | — | — | 1 | 6.11 |
| CHEMBL213212 | — | — | 1 | 5.52 |
| CHEMBL380169 | — | — | 1 | 5.52 |
| CHEMBL379955 | — | — | 1 | 5.30 |
| CHEMBL384592 | — | — | 1 | 5.22 |
| CHEMBL213397 | — | — | 1 | 5.00 |
| CHEMBL384372 | — | — | 1 | - |
| CHEMBL214676 | — | — | 1 | - |
| CHEMBL214586 | — | — | 1 | - |
| CHEMBL379362 | — | — | 1 | - |
| CHEMBL377117 | — | — | 1 | - |
| CHEMBL212348 | — | — | 1 | - |
| CHEMBL216025 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL385537 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL385536 | — | IC50 | = | 39.0 | nM | 7.41 |
| CHEMBL438246 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL214960 | — | IC50 | = | 190.0 | nM | 6.72 |
| CHEMBL385412 | — | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL385156 | — | IC50 | = | 770.0 | nM | 6.11 |
| CHEMBL213212 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL380169 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL379955 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL384592 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL213397 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL384372 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL214676 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL214586 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL379362 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL377117 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL212348 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL216025 | — | IC50 | > | 30000.0 | nM | - |