Assay Detail
Functional
CHEMBL869550
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Competitive inhibition of UGT2B17-catalyzed scopoletin glucuronidation
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Stereochemical sensitivity of the human UDP-glucuronosyltransferases 2B7 and 2B17.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 4.24 | 4.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL206457 | — | — | 1 | 4.24 |
| CHEMBL204019 | — | — | 1 | - |
| CHEMBL202791 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL206457 | — | Ki | = | 57800.0 | nM | 4.24 |
| CHEMBL204019 | — | Ki | = | 201000.0 | nM | - |
| CHEMBL202791 | — | Ki | = | 427000.0 | nM | - |