Assay Detail
Binding
CHEMBL872840
Review assay metadata, readout intent, target linkage, and publication context from the same page.
The compound was evaluated in vitro for the inhibition of Neutral endopeptidase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Asymmetric synthesis of BB-3497--a potent peptide deformylase inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.74 | 5.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL308333 | ACTINONIN | — | 1 | 5.17 |
| CHEMBL431210 | — | — | 1 | 4.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL308333 | ACTINONIN | IC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL431210 | — | IC50 | = | 50000.0 | nM | 4.30 |