Assay Detail
Functional
CHEMBL873918
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The compound tested for agonistic activity against Opioid receptor delta 1 using [3H]- NT1 as the radioligand.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
7-Spiroindanyl derivatives of naltrexone and oxymorphone as selective ligands for delta opioid receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.08 | 9.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL610293 | — | — | 1 | 9.60 |
| CHEMBL399708 | SPIROINDANYLOXYMORPHONE | — | 1 | 8.56 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL610293 | — | Ki | = | 0.25 | nM | 9.60 |
| CHEMBL399708 | SPIROINDANYLOXYMORPHONE | Ki | = | 2.75 | nM | 8.56 |