Assay Detail
Binding
CHEMBL874550
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Inhibitory concentration required against human GLP1 receptor expressed in CHO cell membrane homogenates
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Identification of CJC-1131-albumin bioconjugate as a stable and bioactive GLP-1(7-36) analog.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 9 | 6.53 | 7.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL410972 | — | — | 1 | 7.85 |
| CHEMBL2371792 | — | — | 1 | 7.06 |
| CHEMBL2371793 | — | — | 1 | 6.97 |
| CHEMBL412288 | — | — | 1 | 6.53 |
| CHEMBL409873 | — | — | 1 | 6.34 |
| CHEMBL439104 | — | — | 1 | 6.15 |
| CHEMBL410973 | — | — | 1 | 6.09 |
| CHEMBL265428 | — | — | 1 | 5.27 |
| CHEMBL409371 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL410972 | — | IC50 | = | 14.0 | nM | 7.85 |
| CHEMBL2371792 | — | IC50 | = | 87.0 | nM | 7.06 |
| CHEMBL2371793 | — | IC50 | = | 108.0 | nM | 6.97 |
| CHEMBL412288 | — | IC50 | = | 296.0 | nM | 6.53 |
| CHEMBL409873 | — | IC50 | = | 454.0 | nM | 6.34 |
| CHEMBL439104 | — | IC50 | = | 713.0 | nM | 6.15 |
| CHEMBL410973 | — | IC50 | = | 804.0 | nM | 6.09 |
| CHEMBL265428 | — | IC50 | = | 5354.0 | nM | 5.27 |
| CHEMBL409371 | — | IC50 | > | 10000.0 | nM | - |