Assay Detail
Binding
CHEMBL875000
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of 0.1 nM [3H]pCCK-8 from guinea pig pancreatic membranes
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis and binding affinities of cyclic and related linear analogues of CCK8 selective for central receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.70 | 5.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL273880 | — | — | 1 | 5.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL273880 | — | Ki | = | 1997.0 | nM | 5.70 |