Assay Detail
Binding
CHEMBL875052
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical microsomes.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Angiotensin II receptor antagonists: imidazoles and pyrroles bearing hydroxymethyl and carboxy substituents
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.84 | 7.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL49170 | — | — | 1 | 7.04 |
| CHEMBL274447 | — | — | 1 | 6.64 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL49170 | — | IC50 | = | 92.0 | nM | 7.04 |
| CHEMBL274447 | — | IC50 | = | 230.0 | nM | 6.64 |