Assay Detail
Binding
CHEMBL875190
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Binding affinity against D2L receptor
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Diaminopyrimidine and diaminopyridine 5-HT7 ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 6.43 | 6.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL363452 | — | — | 1 | 6.43 |
| CHEMBL182071 | — | — | 1 | - |
| CHEMBL183277 | — | — | 1 | - |
| CHEMBL183423 | — | — | 1 | - |
| CHEMBL184789 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL363452 | — | Ki | = | 370.0 | nM | 6.43 |
| CHEMBL182071 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL183277 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL183423 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL184789 | — | Ki | > | 1000.0 | nM | - |