Assay Detail
Binding
CHEMBL876365
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Inhibitory constant for Norepinephrine transporter
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of CC chemokine receptor-3 (CCR3) antagonists with picomolar potency.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.04 | 6.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL195433 | — | — | 1 | 6.21 |
| CHEMBL250689 | — | — | 1 | 6.02 |
| CHEMBL363840 | — | — | 1 | 5.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL195433 | — | Ki | = | 611.0 | nM | 6.21 |
| CHEMBL250689 | — | Ki | = | 946.0 | nM | 6.02 |
| CHEMBL363840 | — | Ki | = | 1260.0 | nM | 5.90 |