Assay Detail
Functional
CHEMBL878884
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of cellular growth against mouse (L1210) deficient in thymidine kinase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | L1210 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Design of enzyme inhibitors using iterative protein crystallographic analysis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.37 | 5.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL301423 | — | — | 1 | 5.37 |
| CHEMBL57333 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL301423 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL57333 | — | IC50 | > | 10700.0 | nM | - |