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Assay Detail

CHEMBL880850

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Binding
Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance P
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Substance-P receptor (CHEMBL249)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Identification of L-tryptophan derivatives with potent and selective antagonist activity at the NK1 receptor.
MacLeod AM, Merchant KJ, Brookfield F, Kelleher F, Stevenson G, Owens AP, Swain CJ, Casiceri MA, Sadowski S, Ber E.
J Med Chem (1994) 37 : 1269 -1274
PubMed 7513763 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 31 6.80 9.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL16192 CP-96345 1 9.40
CHEMBL22870 L-732138 1 8.80
CHEMBL282290 1 8.57
CHEMBL278849 L-709400 1 8.10
CHEMBL278351 1 7.66
CHEMBL23926 1 7.52
CHEMBL26336 1 7.21
CHEMBL23129 L-708568 1 7.17
CHEMBL23597 1 7.06
CHEMBL23851 1 6.99
CHEMBL281804 1 6.90
CHEMBL24549 1 6.88
CHEMBL280422 1 6.86
CHEMBL23822 1 6.82
CHEMBL281194 1 6.74
CHEMBL283989 1 6.71
CHEMBL279500 1 6.61
CHEMBL24314 1 6.55
CHEMBL429395 1 6.38
CHEMBL23077 1 6.36
CHEMBL23715 1 6.26
CHEMBL23927 1 6.22
CHEMBL23928 1 6.12
CHEMBL279916 1 5.98
CHEMBL279050 1 5.81
CHEMBL23184 1 5.67
CHEMBL26623 1 5.42
CHEMBL2114308 1 5.26
CHEMBL282728 1 5.26
CHEMBL278555 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL16192 CP-96345 IC50 = 0.4 nM 9.40
CHEMBL22870 L-732138 IC50 = 1.6 nM 8.80
CHEMBL282290 IC50 = 2.7 nM 8.57
CHEMBL278849 L-709400 IC50 = 8.0 nM 8.10
CHEMBL278351 IC50 = 22.0 nM 7.66
CHEMBL23926 IC50 = 30.0 nM 7.52
CHEMBL26336 IC50 = 62.0 nM 7.21
CHEMBL23129 L-708568 IC50 = 67.0 nM 7.17
CHEMBL23597 IC50 = 87.0 nM 7.06
CHEMBL23851 IC50 = 103.0 nM 6.99
CHEMBL281804 IC50 = 125.0 nM 6.90
CHEMBL24549 IC50 = 133.0 nM 6.88
CHEMBL280422 IC50 = 138.0 nM 6.86
CHEMBL23822 IC50 = 153.0 nM 6.82
CHEMBL281194 IC50 = 183.0 nM 6.74
CHEMBL283989 IC50 = 197.0 nM 6.71
CHEMBL279500 IC50 = 243.0 nM 6.61
CHEMBL24314 IC50 = 280.0 nM 6.55
CHEMBL429395 IC50 = 413.0 nM 6.38
CHEMBL23077 IC50 = 433.0 nM 6.36
CHEMBL23715 IC50 = 553.0 nM 6.26
CHEMBL23927 IC50 = 600.0 nM 6.22
CHEMBL23928 IC50 = 760.0 nM 6.12
CHEMBL279916 IC50 = 1050.0 nM 5.98
CHEMBL279050 IC50 = 1533.0 nM 5.81
CHEMBL23184 IC50 = 2150.0 nM 5.67
CHEMBL26623 IC50 = 3800.0 nM 5.42
CHEMBL2114308 IC50 = 5500.0 nM 5.26
CHEMBL282728 IC50 = 5500.0 nM 5.26
CHEMBL278555 IC50 > 10000.0 nM -
CHEMBL279915 IC50 > 100.0 nM -