Assay Detail
Binding
CHEMBL881284
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Effective concentration required for binding to wild-type TAR using electrophoretic mobility shift assays done at at 25 degree C with pH 7.5
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human immunodeficiency virus 1 |
| Confidence | 3 — Cell-line / Tissue |
| Curated By | Expert |
Publication
Antiviral 6-amino-quinolones: molecular basis for potency and selectivity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 6.72 | 6.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL188588 | — | — | 1 | 6.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL188588 | — | EC50 | = | 190.0 | nM | 6.72 |