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Assay Detail

CHEMBL881599

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested for inhibition of bovine beta trypsin
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Bos taurus
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Trypsin-3 (CHEMBL4551)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis and evaluation of the sunflower derived trypsin inhibitor as a potent inhibitor of the type II transmembrane serine protease, matriptase.
Long YQ, Lee SL, Lin CY, Enyedy IJ, Wang S, Li P, Dickson RB, Roller PP.
Bioorg Med Chem Lett (2001) 11 : 2515 -2519
PubMed 11549459 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.97 8.97

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL239127 1 8.97

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL239127 Ki = 1.06 nM 8.97