Assay Detail
Binding
CHEMBL881769
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Inhibitory concentration against angiotensin II receptor, type 2
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Designed multiple ligands. An emerging drug discovery paradigm.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.33 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL302102 | — | — | 1 | 9.15 |
| CHEMBL372814 | — | — | 1 | 7.50 |
| CHEMBL24322 | — | — | 1 | 5.35 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL302102 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL372814 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL24322 | — | IC50 | = | 4500.0 | nM | 5.35 |