Assay Detail
Binding
CHEMBL884356
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Compound was tested for its inhibitory activity against cyclin-dependent kinase 5
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
3D-QSAR CoMFA on cyclin-dependent kinase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.35 | 6.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL422759 | — | — | 1 | 6.40 |
| CHEMBL25840 | — | — | 1 | 6.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL422759 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL25840 | — | IC50 | = | 500.0 | nM | 6.30 |