Assay Detail
Binding
CHEMBL884735
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory constant against the protein kinase A
6
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Target
cAMP-dependent protein kinase (PKA) (CHEMBL2094138) ↗| Type | PROTEIN FAMILY |
| Organism | Homo sapiens |
Publication
Joys of molecules. 2. Endeavors in chemical biology and medicinal chemistry.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 6 | 8.40 | 8.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL365598 | — | — | 2 | 8.47 |
| CHEMBL193697 | — | — | 2 | 8.41 |
| CHEMBL60254 | BALANOL | — | 2 | 8.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL365598 | — | Ki | = | 3.4 | nM | 8.47 |
| CHEMBL365598 | — | Ki | = | 3.4 | nM | 8.47 |
| CHEMBL193697 | — | Ki | = | 3.9 | nM | 8.41 |
| CHEMBL193697 | — | Ki | = | 3.9 | nM | 8.41 |
| CHEMBL60254 | BALANOL | Ki | = | 4.7 | nM | 8.33 |
| CHEMBL60254 | BALANOL | Ki | = | 4.7 | nM | 8.33 |