Assay Detail
Functional
CHEMBL886395
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Inhibition EGF-dependent mitogenesis of mouse BaF/ERX cells by [3H]thymidine incorporation assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | BaF/ERX |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and biological evaluation of analogues of the anti-tumor alkaloid naamidine A.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 4.82 | 5.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL339727 | — | — | 1 | 5.52 |
| CHEMBL246293 | — | — | 1 | 5.40 |
| CHEMBL397390 | — | — | 1 | 5.30 |
| CHEMBL247533 | — | — | 1 | 5.00 |
| CHEMBL245882 | — | — | 1 | 4.92 |
| CHEMBL393225 | — | — | 1 | 4.82 |
| CHEMBL246294 | — | — | 1 | 4.75 |
| CHEMBL247729 | — | — | 1 | 4.60 |
| CHEMBL247532 | — | — | 1 | 4.30 |
| CHEMBL397333 | — | — | 1 | 4.30 |
| CHEMBL246083 | NAAMINE A | — | 1 | 4.12 |
| CHEMBL247129 | — | — | 1 | - |
| CHEMBL394400 | — | — | 1 | - |
| CHEMBL247534 | — | — | 1 | - |
| CHEMBL247334 | — | — | 1 | - |
| CHEMBL245681 | — | — | 1 | - |
| CHEMBL245486 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL339727 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL246293 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL397390 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL247533 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL245882 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL393225 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL246294 | — | IC50 | = | 18000.0 | nM | 4.75 |
| CHEMBL247729 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL247532 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL397333 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL246083 | NAAMINE A | IC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL247129 | — | IC50 | > | 75000.0 | nM | - |
| CHEMBL394400 | — | IC50 | > | 75000.0 | nM | - |
| CHEMBL247534 | — | IC50 | > | 75000.0 | nM | - |
| CHEMBL247334 | — | IC50 | > | 75000.0 | nM | - |
| CHEMBL245681 | — | IC50 | > | 75000.0 | nM | - |
| CHEMBL245486 | — | IC50 | > | 75000.0 | nM | - |