Assay Detail
Binding
CHEMBL886478
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Activity at RXRalpha by GAL4DNA cotransfection assay
20
Total Activities
20
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
RXR-LXR heterodimer modulators for the potential treatment of dyslipidemia.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 19 | 7.56 | 9.05 |
| Activity | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL248415 | — | — | 1 | 9.05 |
| CHEMBL246821 | — | — | 1 | 8.74 |
| CHEMBL247005 | — | — | 1 | 8.74 |
| CHEMBL246629 | — | — | 1 | 8.68 |
| CHEMBL428930 | — | — | 1 | 7.79 |
| CHEMBL247819 | — | — | 1 | 7.74 |
| CHEMBL247836 | — | — | 1 | 7.61 |
| CHEMBL248191 | — | — | 1 | 7.21 |
| CHEMBL400557 | — | — | 1 | 7.17 |
| CHEMBL247012 | — | — | 1 | 7.01 |
| CHEMBL247856 | — | — | 1 | 6.76 |
| CHEMBL400380 | — | — | 1 | 5.92 |
| CHEMBL247011 | — | — | 1 | 5.80 |
| CHEMBL247855 | — | — | 1 | - |
| CHEMBL246805 | — | — | 1 | - |
| CHEMBL399765 | — | — | 1 | - |
| CHEMBL247857 | — | — | 1 | - |
| CHEMBL400490 | — | — | 1 | - |
| CHEMBL246625 | — | — | 1 | - |
| CHEMBL246806 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL248415 | — | EC50 | = | 0.9 | nM | 9.05 |
| CHEMBL246821 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL247005 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL246629 | — | EC50 | = | 2.1 | nM | 8.68 |
| CHEMBL428930 | — | EC50 | = | 16.3 | nM | 7.79 |
| CHEMBL247819 | — | EC50 | = | 18.3 | nM | 7.74 |
| CHEMBL247836 | — | EC50 | = | 24.3 | nM | 7.61 |
| CHEMBL248191 | — | EC50 | = | 61.2 | nM | 7.21 |
| CHEMBL400557 | — | EC50 | = | 67.3 | nM | 7.17 |
| CHEMBL247012 | — | EC50 | = | 96.6 | nM | 7.01 |
| CHEMBL247856 | — | EC50 | = | 173.1 | nM | 6.76 |
| CHEMBL400380 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL247011 | — | EC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL247855 | — | EC50 | - | — | - | |
| CHEMBL246805 | — | EC50 | - | — | - | |
| CHEMBL399765 | — | Activity | - | — | - | |
| CHEMBL247857 | — | EC50 | - | — | - | |
| CHEMBL400490 | — | EC50 | - | — | - | |
| CHEMBL246625 | — | EC50 | - | — | - | |
| CHEMBL246806 | — | EC50 | > | 10000.0 | nM | - |