Assay Detail
Functional
CHEMBL887763
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Antimicrobial activity against Plasmodium falciparum in erythrocytes
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Additional interaction of allophenylnorstatine-containing tripeptidomimetics with malarial aspartic protease plasmepsin II.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 5.34 | 5.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL440965 | — | — | 1 | 5.51 |
| CHEMBL411559 | — | — | 1 | 5.33 |
| CHEMBL231522 | — | — | 1 | 5.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL440965 | — | EC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL411559 | — | EC50 | = | 4700.0 | nM | 5.33 |
| CHEMBL231522 | — | EC50 | = | 6800.0 | nM | 5.17 |