Assay Detail
Binding
CHEMBL888093
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Binding affinity to human recombinant sst4 receptor
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Identification and SAR of potent and selective non-peptide obeline somatostatin sst1 receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| pKd | 2 | - | - |
| Kd | 1 | 4.82 | 4.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL251541 | OBELIN | — | 1 | 4.82 |
| CHEMBL249113 | — | — | 1 | - |
| CHEMBL249112 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL251541 | OBELIN | Kd | = | 15135.61 | nM | 4.82 |
| CHEMBL249113 | — | pKd | - | — | - | |
| CHEMBL249112 | — | pKd | - | — | - |