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Assay Detail

CHEMBL896739

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against mouse L1210 cells by MTT assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type L1210
Confidence 1 — Organism
Curated By Autocuration

Target

L1210 (CHEMBL386)
Type CELL-LINE
Organism Mus musculus

Publication

Synthesis and bioevaluation of N-(arylalkyl)-homospermidine conjugates.
Xie S, Cheng P, Liu G, Ma Y, Zhao J, Chehtane M, Khaled AR, Phanstiel O, Wang C.
Bioorg Med Chem Lett (2007) 17 : 4471 -4475
PubMed 17574415 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 4.87 5.32

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL540552 1 5.32
CHEMBL540336 1 5.09
CHEMBL536076 1 5.00
CHEMBL536297 1 4.83
CHEMBL536524 1 4.82
CHEMBL557367 1 4.82
CHEMBL536075 1 4.77
CHEMBL536525 1 4.69
CHEMBL536523 1 4.45
CHEMBL536299 1 -
CHEMBL540379 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL540552 IC50 = 4800.0 nM 5.32
CHEMBL540336 IC50 = 8040.0 nM 5.09
CHEMBL536076 IC50 = 9980.0 nM 5.00
CHEMBL536297 IC50 = 14770.0 nM 4.83
CHEMBL536524 IC50 = 15090.0 nM 4.82
CHEMBL557367 IC50 = 15060.0 nM 4.82
CHEMBL536075 IC50 = 16940.0 nM 4.77
CHEMBL536525 IC50 = 20260.0 nM 4.69
CHEMBL536523 IC50 = 35770.0 nM 4.45
CHEMBL536299 IC50 > 50000.0 nM -
CHEMBL540379 IC50 > 50000.0 nM -