Assay Detail
Functional
CHEMBL897415
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Antiviral activity against HCV in Huh7-Rep cells by luciferase assay
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Hepacivirus hominis |
| Cell Type | Huh7-Rep |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Evaluation of the anti-hepatitis C virus effect of novel potent, selective, and orally bioavailable JNK and VEGFR kinase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 31 | 5.82 | 7.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL234655 | — | — | 1 | 7.19 |
| CHEMBL237476 | — | — | 1 | 7.08 |
| CHEMBL235131 | — | — | 1 | 6.46 |
| CHEMBL237684 | — | — | 1 | 6.26 |
| CHEMBL401035 | — | — | 1 | 6.23 |
| CHEMBL235129 | — | — | 1 | 6.15 |
| CHEMBL234652 | — | — | 1 | 6.10 |
| CHEMBL237902 | — | — | 1 | 6.07 |
| CHEMBL238125 | — | — | 1 | 6.05 |
| CHEMBL237477 | — | — | 1 | 6.04 |
| CHEMBL234481 | — | — | 1 | 6.00 |
| CHEMBL237903 | — | — | 1 | 6.00 |
| CHEMBL237046 | — | — | 1 | 5.92 |
| CHEMBL238334 | — | — | 1 | 5.78 |
| CHEMBL238127 | — | — | 1 | 5.72 |
| CHEMBL234651 | — | — | 1 | 5.71 |
| CHEMBL399011 | — | — | 1 | 5.70 |
| CHEMBL401016 | — | — | 1 | 5.70 |
| CHEMBL234480 | — | — | 1 | 5.66 |
| CHEMBL401034 | — | — | 1 | 5.60 |
| CHEMBL237265 | — | — | 1 | 5.58 |
| CHEMBL236837 | — | — | 1 | 5.44 |
| CHEMBL234478 | — | — | 1 | 5.44 |
| CHEMBL234653 | — | — | 1 | 5.44 |
| CHEMBL235350 | — | — | 1 | 5.40 |
| CHEMBL442241 | — | — | 1 | 5.34 |
| CHEMBL392307 | — | — | 1 | 5.30 |
| CHEMBL391448 | — | — | 1 | 5.19 |
| CHEMBL237686 | — | — | 1 | 5.02 |
| CHEMBL439034 | — | — | 1 | 5.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL234655 | — | EC50 | = | 64.0 | nM | 7.19 |
| CHEMBL237476 | — | EC50 | = | 84.0 | nM | 7.08 |
| CHEMBL235131 | — | EC50 | = | 350.0 | nM | 6.46 |
| CHEMBL237684 | — | EC50 | = | 550.0 | nM | 6.26 |
| CHEMBL401035 | — | EC50 | = | 590.0 | nM | 6.23 |
| CHEMBL235129 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL234652 | — | EC50 | = | 800.0 | nM | 6.10 |
| CHEMBL237902 | — | EC50 | = | 850.0 | nM | 6.07 |
| CHEMBL238125 | — | EC50 | = | 890.0 | nM | 6.05 |
| CHEMBL237477 | — | EC50 | = | 920.0 | nM | 6.04 |
| CHEMBL234481 | — | EC50 | = | 990.0 | nM | 6.00 |
| CHEMBL237903 | — | EC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL237046 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL238334 | — | EC50 | = | 1670.0 | nM | 5.78 |
| CHEMBL238127 | — | EC50 | = | 1910.0 | nM | 5.72 |
| CHEMBL234651 | — | EC50 | = | 1960.0 | nM | 5.71 |
| CHEMBL399011 | — | EC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL401016 | — | EC50 | = | 1980.0 | nM | 5.70 |
| CHEMBL234480 | — | EC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL401034 | — | EC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL237265 | — | EC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL236837 | — | EC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL234478 | — | EC50 | = | 3650.0 | nM | 5.44 |
| CHEMBL234653 | — | EC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL235350 | — | EC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL442241 | — | EC50 | = | 4600.0 | nM | 5.34 |
| CHEMBL392307 | — | EC50 | = | 4950.0 | nM | 5.30 |
| CHEMBL391448 | — | EC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL237686 | — | EC50 | = | 9600.0 | nM | 5.02 |
| CHEMBL439034 | — | EC50 | = | 9950.0 | nM | 5.00 |
| CHEMBL395587 | — | EC50 | > | 50000.0 | nM | - |