Assay Detail
Functional
CHEMBL901902
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Inhibition of IgE production in antigen-sensitized BALB/c mouse spleen cells
24
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Tissue | Spleen |
| Cell Type | spleen |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
2-phenylimidazopyridines, a new series of Golgi compounds with potent antiviral activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 24 | 8.21 | 9.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL238471 | — | — | 1 | 9.82 |
| CHEMBL239543 | — | — | 1 | 9.82 |
| CHEMBL239542 | — | — | 1 | 9.00 |
| CHEMBL395450 | — | — | 1 | 9.00 |
| CHEMBL223973 | — | — | 1 | 9.00 |
| CHEMBL397884 | — | — | 1 | 9.00 |
| CHEMBL239335 | — | — | 1 | 8.82 |
| CHEMBL397173 | — | — | 1 | 8.52 |
| CHEMBL238469 | — | — | 1 | 8.52 |
| CHEMBL240134 | — | — | 1 | 8.40 |
| CHEMBL222659 | — | — | 2 | 8.40 |
| CHEMBL373757 | — | — | 1 | 8.30 |
| CHEMBL240389 | — | — | 1 | 8.30 |
| CHEMBL393953 | — | — | 1 | 8.00 |
| CHEMBL241197 | — | — | 1 | 8.00 |
| CHEMBL3085094 | — | — | 1 | 8.00 |
| CHEMBL240133 | — | — | 1 | 8.00 |
| CHEMBL273339 | — | — | 1 | 8.00 |
| CHEMBL395451 | — | — | 1 | 7.35 |
| CHEMBL375891 | — | — | 1 | 7.16 |
| CHEMBL238906 | — | — | 1 | 6.92 |
| CHEMBL397885 | — | — | 1 | 6.85 |
| CHEMBL240596 | — | — | 1 | 6.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL238471 | — | IC50 | = | 0.15 | nM | 9.82 |
| CHEMBL239543 | — | IC50 | = | 0.15 | nM | 9.82 |
| CHEMBL239542 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL223973 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL397884 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL395450 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL239335 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL397173 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL238469 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL240134 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL222659 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL373757 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL240389 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL240133 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL273339 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL3085094 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL241197 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL393953 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL222659 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL395451 | — | IC50 | = | 45.0 | nM | 7.35 |
| CHEMBL375891 | — | IC50 | = | 70.0 | nM | 7.16 |
| CHEMBL238906 | — | IC50 | = | 120.0 | nM | 6.92 |
| CHEMBL397885 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL240596 | — | IC50 | = | 1000.0 | nM | 6.00 |