Assay Detail
Binding
CHEMBL906657
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant deoxyhypusine synthase in Plasmodium falciparum NF54
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Plasmodium falciparum NF54 |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Modification of eukaryotic initiation factor 5A from Plasmodium vivax by a truncated deoxyhypusine synthase from Plasmodium falciparum: An enzyme with dual enzymatic properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.65 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL229457 | — | — | 1 | 7.00 |
| CHEMBL28242 | — | — | 1 | 4.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL229457 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL28242 | — | Ki | = | 50000.0 | nM | 4.30 |