Assay Detail
Binding
CHEMBL914209
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Inhibition of Aspergillus nidulans RmtA by TRF assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Aspergillus nidulans |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Target-based approach to inhibitors of histone arginine methyltransferases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.69 | 5.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL227725 | ALLANTODAPSONE | — | 1 | 5.08 |
| CHEMBL142304 | STILBAMIDINE | 2.0 | 1 | 4.52 |
| CHEMBL221047 | — | — | 1 | 4.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL227725 | ALLANTODAPSONE | IC50 | = | 8300.0 | nM | 5.08 |
| CHEMBL142304 | STILBAMIDINE | IC50 | = | 29900.0 | nM | 4.52 |
| CHEMBL221047 | — | IC50 | = | 33800.0 | nM | 4.47 |