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Assay Detail

CHEMBL914291

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Functional
Antiparasitic activity against chloroquine-resistant Plasmodium falciparum ItG after 48 hrs by SYBR-Green assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Intermediate

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

A potent, covalent inhibitor of orotidine 5'-monophosphate decarboxylase with antimalarial activity.
Bello AM, Poduch E, Fujihashi M, Amani M, Li Y, Crandall I, Hui R, Lee PI, Kain KC, Pai EF, Kotra LP.
J Med Chem (2007) 50 : 915 -921
PubMed 17290979 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.36 5.36

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL220442 1 5.36

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL220442 IC50 = 4400.0 nM 5.36