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Assay Detail

CHEMBL916302

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of COX2 in human whole blood assessed as inhibition of LPS-stimulated PGE2 production
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Tissue Blood
Confidence 9 — Direct single protein target
Curated By Intermediate

Target

Prostaglandin G/H synthase 2 (CHEMBL230)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Design, synthesis, and pharmacological evaluation of pyridinic analogues of nimesulide as cyclooxygenase-2 selective inhibitors.
Julémont F, de Leval X, Michaux C, Renard JF, Winum JY, Montero JL, Damas J, Dogné JM, Pirotte B.
J Med Chem (2004) 47 : 6749 -6759
PubMed 15615524 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 29 5.87 7.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL224400 1 7.05
CHEMBL224136 1 6.92
CHEMBL388628 1 6.89
CHEMBL224640 1 6.82
CHEMBL118 CELECOXIB 4.0 1 6.46
CHEMBL225092 1 6.36
CHEMBL224612 1 6.28
CHEMBL147165 1 6.21
CHEMBL56367 NIMESULIDE 4.0 1 6.16
CHEMBL224122 1 5.92
CHEMBL225113 1 5.82
CHEMBL388625 1 5.73
CHEMBL224192 1 5.70
CHEMBL224624 1 5.63
CHEMBL387879 1 5.59
CHEMBL223655 1 5.48
CHEMBL224193 1 5.12
CHEMBL374169 1 5.01
CHEMBL374168 1 4.86
CHEMBL376143 1 4.85
CHEMBL224401 1 4.32
CHEMBL224781 1 -
CHEMBL225236 1 -
CHEMBL389485 1 -
CHEMBL224256 1 -
CHEMBL224693 1 -
CHEMBL224201 1 -
CHEMBL148542 1 -
CHEMBL390317 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL224400 IC50 = 90.0 nM 7.05
CHEMBL224136 IC50 = 120.0 nM 6.92
CHEMBL388628 IC50 = 130.0 nM 6.89
CHEMBL224640 IC50 = 150.0 nM 6.82
CHEMBL118 CELECOXIB IC50 = 350.0 nM 6.46
CHEMBL225092 IC50 = 440.0 nM 6.36
CHEMBL224612 IC50 = 530.0 nM 6.28
CHEMBL147165 IC50 = 620.0 nM 6.21
CHEMBL56367 NIMESULIDE IC50 = 700.0 nM 6.16
CHEMBL224122 IC50 = 1190.0 nM 5.92
CHEMBL225113 IC50 = 1530.0 nM 5.82
CHEMBL388625 IC50 = 1870.0 nM 5.73
CHEMBL224192 IC50 = 1990.0 nM 5.70
CHEMBL224624 IC50 = 2360.0 nM 5.63
CHEMBL387879 IC50 = 2550.0 nM 5.59
CHEMBL223655 IC50 = 3280.0 nM 5.48
CHEMBL224193 IC50 = 7600.0 nM 5.12
CHEMBL374169 IC50 = 9690.0 nM 5.01
CHEMBL374168 IC50 = 13840.0 nM 4.86
CHEMBL376143 IC50 = 14110.0 nM 4.85
CHEMBL224401 IC50 = 47620.0 nM 4.32
CHEMBL224781 IC50 > 100000.0 nM -
CHEMBL225236 IC50 > 100000.0 nM -
CHEMBL389485 IC50 > 100000.0 nM -
CHEMBL224256 IC50 > 100000.0 nM -
CHEMBL224693 IC50 > 100000.0 nM -
CHEMBL224201 IC50 > 100000.0 nM -
CHEMBL148542 IC50 > 100000.0 nM -
CHEMBL390317 IC50 > 100000.0 nM -