Assay Detail
Functional
CHEMBL916350
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Effect on modulating pentamidine-resistance of Leishmania enriettii LePentR50 assessed as decrease in survival after 72 hrs by MTS
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Flavonoid dimers as bivalent modulators for pentamidine and sodium stiboglucanate resistance in leishmania.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.88 | 6.03 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL214738 | — | — | 1 | 6.03 |
| CHEMBL215017 | — | — | 1 | 5.73 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL214738 | — | EC50 | = | 940.0 | nM | 6.03 |
| CHEMBL215017 | — | EC50 | = | 1850.0 | nM | 5.73 |