Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL918816

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human PC3 cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type PC-3
Confidence 1 — Organism
Curated By Autocuration

Target

PC-3 (CHEMBL390)
Type CELL-LINE
Organism Homo sapiens

Publication

In vitro cytotoxicity evaluation of some substituted isatin derivatives.
Vine KL, Locke JM, Ranson M, Benkendorff K, Pyne SG, Bremner JB.
Bioorg Med Chem (2007) 15 : 931 -938
PubMed 17088067 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 4.37 4.59

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL376616 1 4.59
CHEMBL388580 1 4.39
CHEMBL387839 1 4.14
CHEMBL388579 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL376616 IC50 = 25900.0 nM 4.59
CHEMBL388580 IC50 = 41000.0 nM 4.39
CHEMBL387839 IC50 = 71900.0 nM 4.14
CHEMBL388579 IC50 = 101000.0 nM -