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Assay Detail

CHEMBL920546

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to HCV 40-mer RNA by MS based binding assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Hepacivirus hominis
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

SAR by MS: discovery of a new class of RNA-binding small molecules for the hepatitis C virus: internal ribosome entry site IIA subdomain.
Seth PP, Miyaji A, Jefferson EA, Sannes-Lowery KA, Osgood SA, Propp SS, Ranken R, Massire C, Sampath R, Ecker DJ, Swayze EE, Griffey RH.
J Med Chem (2005) 48 : 7099 -7102
PubMed 16279767 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 6 5.64 6.14

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL223720 1 6.14
CHEMBL223608 1 6.07
CHEMBL388502 1 5.77
CHEMBL224788 1 5.46
CHEMBL224999 1 4.77
CHEMBL427101 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL223720 Kd = 720.0 nM 6.14
CHEMBL223608 Kd = 860.0 nM 6.07
CHEMBL388502 Kd = 1700.0 nM 5.77
CHEMBL224788 Kd = 3500.0 nM 5.46
CHEMBL224999 Kd = 17000.0 nM 4.77
CHEMBL427101 Kd > 100000.0 nM -