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Assay Detail

CHEMBL920547

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Functional
Reduction of HCV RNA levels by HCV replicon assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Intermediate

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

SAR by MS: discovery of a new class of RNA-binding small molecules for the hepatitis C virus: internal ribosome entry site IIA subdomain.
Seth PP, Miyaji A, Jefferson EA, Sannes-Lowery KA, Osgood SA, Propp SS, Ranken R, Massire C, Sampath R, Ecker DJ, Swayze EE, Griffey RH.
J Med Chem (2005) 48 : 7099 -7102
PubMed 16279767 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 6 5.09 5.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL388502 1 5.82
CHEMBL223608 1 5.41
CHEMBL223720 1 5.27
CHEMBL224788 1 4.54
CHEMBL224999 1 4.43
CHEMBL427101 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL388502 EC50 = 1500.0 nM 5.82
CHEMBL223608 EC50 = 3900.0 nM 5.41
CHEMBL223720 EC50 = 5400.0 nM 5.27
CHEMBL224788 EC50 = 29000.0 nM 4.54
CHEMBL224999 EC50 = 37000.0 nM 4.43
CHEMBL427101 EC50 - -