Assay Detail
Functional
CHEMBL921073
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antitumor activity against human HepG2 cells
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HepG2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | - | - |
| EC50 | 1 | 5.68 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL437612 | — | — | 1 | 5.68 |
| CHEMBL290904 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL437612 | — | EC50 | = | 2070.0 | nM | 5.68 |
| CHEMBL290904 | — | IC50 | = | 1210.0 | ug.mL-1 | - |