Assay Detail
Binding
CHEMBL922325
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of adrenergic alpha 1 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and structure-affinity relationships of novel spirocyclic sigma receptor ligands with furopyrazole structure.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.91 | 5.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL259732 | — | — | 1 | 5.91 |
| CHEMBL410832 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL259732 | — | IC50 | = | 1218.0 | nM | 5.91 |
| CHEMBL410832 | — | IC50 | > | 1000.0 | nM | - |