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Assay Detail

CHEMBL923030

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human PC3 cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type PC-3
Confidence 1 — Organism
Curated By Autocuration

Target

PC-3 (CHEMBL390)
Type CELL-LINE
Organism Homo sapiens

Publication

N-phenethyl and N-naphthylmethyl isatins and analogues as in vitro cytotoxic agents.
Matesic L, Locke JM, Bremner JB, Pyne SG, Skropeta D, Ranson M, Vine KL.
Bioorg Med Chem (2008) 16 : 3118 -3124
PubMed 18182300 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.71 5.84

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL406943 1 5.84
CHEMBL406631 1 5.68
CHEMBL406207 1 5.66
CHEMBL260493 1 5.64

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL406943 IC50 = 1440.0 nM 5.84
CHEMBL406631 IC50 = 2090.0 nM 5.68
CHEMBL406207 IC50 = 2210.0 nM 5.66
CHEMBL260493 IC50 = 2290.0 nM 5.64