Assay Detail
Binding
CHEMBL923901
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Inhibition of PDGFR expressed in NIH cells by Western blot analysis
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | NIH |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Formation of fluorine-18 labeled diaryl ureas--labeled VEGFR-2/PDGFR dual inhibitors as molecular imaging agents for angiogenesis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 8.70 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL259394 | — | — | 1 | 8.70 |
| CHEMBL179815 | — | — | 1 | 8.70 |
| CHEMBL259395 | — | — | 1 | 8.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL259394 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL179815 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL259395 | — | IC50 | = | 2.0 | nM | 8.70 |