Assay Detail
Binding
CHEMBL924919
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Arthrobacter protophormiae endo-beta-N-acetylglucosaminidase after 5 mins by HPAEC-PED method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Arthrobacter protophormiae |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Endo-beta-N-acetylglucosaminidase (CHEMBL1075042) ↗| Type | SINGLE PROTEIN |
| Organism | Arthrobacter protophormiae |
Publication
Synthesis and inhibitory activity of oligosaccharide thiazolines as a class of mechanism-based inhibitors for endo-beta-N-acetylglucosaminidases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.32 | 6.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL259756 | — | — | 1 | 6.66 |
| CHEMBL261523 | — | — | 1 | 4.89 |
| CHEMBL260584 | — | — | 1 | 4.42 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL259756 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL261523 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL260584 | — | IC50 | = | 38000.0 | nM | 4.42 |