Assay Detail
Binding
CHEMBL924920
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Inhibition of Mucor hiemalis endo-beta-N-acetylglucosaminidase after 5 mins by HPAEC-PED method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mucor hiemalis |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and inhibitory activity of oligosaccharide thiazolines as a class of mechanism-based inhibitors for endo-beta-N-acetylglucosaminidases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.50 | 5.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL259756 | — | — | 1 | 5.22 |
| CHEMBL261523 | — | — | 1 | 4.19 |
| CHEMBL260584 | — | — | 1 | 4.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL259756 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL261523 | — | IC50 | = | 64000.0 | nM | 4.19 |
| CHEMBL260584 | — | IC50 | = | 80000.0 | nM | 4.10 |