Assay Detail
Binding
CHEMBL925072
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of 5HT2A receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
CC chemokine receptor-3 (CCR3) antagonists: improving the selectivity of DPC168 by reducing central ring lipophilicity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.66 | 6.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL250689 | — | — | 1 | 6.04 |
| CHEMBL249854 | — | — | 1 | 5.28 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL250689 | — | IC50 | = | 920.0 | nM | 6.04 |
| CHEMBL249854 | — | IC50 | = | 5300.0 | nM | 5.28 |