Assay Detail
Functional
CHEMBL925550
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Antiproliferative activity against human SK-N-MC cells by MTT assay
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SK-N-MC |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Investigating the antiproliferative activity of quinoline-5,8-diones and styrylquinolinecarboxylic acids on tumor cell lines.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 29 | 5.37 | 5.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL388378 | — | — | 1 | 5.37 |
| CHEMBL202312 | — | — | 1 | - |
| CHEMBL402271 | — | — | 1 | - |
| CHEMBL428230 | — | — | 1 | - |
| CHEMBL249172 | — | — | 1 | - |
| CHEMBL249171 | — | — | 1 | - |
| CHEMBL248968 | — | — | 1 | - |
| CHEMBL402270 | — | — | 1 | - |
| CHEMBL248967 | — | — | 1 | - |
| CHEMBL248966 | — | — | 1 | - |
| CHEMBL402269 | — | — | 1 | - |
| CHEMBL248965 | — | — | 1 | - |
| CHEMBL400150 | — | — | 1 | - |
| CHEMBL248772 | — | — | 1 | - |
| CHEMBL248771 | — | — | 1 | - |
| CHEMBL225640 | — | — | 1 | - |
| CHEMBL248769 | — | — | 1 | - |
| CHEMBL400149 | — | — | 1 | - |
| CHEMBL250670 | — | — | 1 | - |
| CHEMBL250487 | — | — | 1 | - |
| CHEMBL446454 | — | — | 1 | - |
| CHEMBL250486 | — | — | 1 | - |
| CHEMBL241898 | — | — | 1 | - |
| CHEMBL250485 | — | — | 1 | - |
| CHEMBL250484 | — | — | 1 | - |
| CHEMBL224238 | — | — | 1 | - |
| CHEMBL250659 | — | — | 1 | - |
| CHEMBL224482 | — | — | 1 | - |
| CHEMBL248770 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL388378 | — | IC50 | = | 4260.0 | nM | 5.37 |
| CHEMBL202312 | — | IC50 | - | — | - | |
| CHEMBL402271 | — | IC50 | - | — | - | |
| CHEMBL428230 | — | IC50 | - | — | - | |
| CHEMBL249172 | — | IC50 | - | — | - | |
| CHEMBL249171 | — | IC50 | - | — | - | |
| CHEMBL248968 | — | IC50 | - | — | - | |
| CHEMBL402270 | — | IC50 | - | — | - | |
| CHEMBL248967 | — | IC50 | - | — | - | |
| CHEMBL248966 | — | IC50 | - | — | - | |
| CHEMBL402269 | — | IC50 | - | — | - | |
| CHEMBL248965 | — | IC50 | - | — | - | |
| CHEMBL400150 | — | IC50 | - | — | - | |
| CHEMBL248772 | — | IC50 | - | — | - | |
| CHEMBL248771 | — | IC50 | - | — | - | |
| CHEMBL225640 | — | IC50 | - | — | - | |
| CHEMBL248769 | — | IC50 | - | — | - | |
| CHEMBL400149 | — | IC50 | - | — | - | |
| CHEMBL250670 | — | IC50 | - | — | - | |
| CHEMBL250487 | — | IC50 | - | — | - | |
| CHEMBL446454 | — | IC50 | - | — | - | |
| CHEMBL250486 | — | IC50 | - | — | - | |
| CHEMBL241898 | — | IC50 | > | 6250.0 | nM | - |
| CHEMBL250485 | — | IC50 | - | — | - | |
| CHEMBL250484 | — | IC50 | - | — | - | |
| CHEMBL224238 | — | IC50 | - | — | - | |
| CHEMBL250659 | — | IC50 | - | — | - | |
| CHEMBL224482 | — | IC50 | > | 6250.0 | nM | - |
| CHEMBL248770 | — | IC50 | - | — | - |