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Assay Detail

CHEMBL926005

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of free prothrombinase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Structure-activity relationships of anthranilamide-based factor Xa inhibitors containing piperidinone and pyridinone P4 moieties.
Corte JR, Fang T, Pinto DJ, Han W, Hu Z, Jiang XJ, Li YL, Gauuan JF, Hadden M, Orton D, Rendina AR, Luettgen JM, Wong PC, He K, Morin PE, Chang CH, Cheney DL, Knabb RM, Wexler RR, Lam PY.
Bioorg Med Chem Lett (2008) 18 : 2845 -2849
PubMed 18424044 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.22 9.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL260085 1 9.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL260085 Ki = 0.6 nM 9.22